2018.06-2020.06,四川大学华西医学院客座副教授;
JACS,Nature Communications, Science Translational Medicien,J. Med. Chem.,Advanced Science 等杂志审稿人。
气体信使小分子(CO, H2S等)药物化学生物学研究:发展新颖的脱笼(decaging)化学,用于气体信使小分子的可控靶向递送,并研究其在相关重大疾病的发生、发展以及治疗方面的作用。
新型Click化学的发现及其相关化学生物学研究:发展新颖的Click反应,并用于相关化学生物学研究,包括生物正交前药的设计,生物大分子的可逆可视化标记等。
抗感染、抗肿瘤靶向小分子药物的设计合成:基于传统药物化学策略,进行抗感染、抗肿瘤小分子靶向药物的设计与合成。
药学(药物化学)学硕,药学专硕,药学/化学生物学博士
Shunfei Cui, # Yiyao Pan, # Chenzhe Ma, Bin Qi, Qingqiang Min, Ming Li, Huabing Chen, * Hengte Ke,* and Xingyue Ji*. Self-assembled carbon monoxide nanoprodrug for chemiexcitation-triggered synergistic chemotherapy against breast cancer. Sci. China Chem., 2025, doi: 10.1007/s11426-024-2465-9.
Jiekai Sun, Xu Wang, Ye Gao, Shuangyu Li, Ziwei Hu, Yan Huang, Baoqiang Fan, Xia Wang, Miao Liu, Chunhua Qiao, Wei Zhang*, Yipeng Wang*, Xingyue Ji*. H2S scavenger as a broad-spectrum strategy to deplete bacteria-derived H2S for antibacterial sensitization. Nat. Commun., 2024, 15, 9422.
Zhicheng Yan, Yiyao Pan, Guofeng Jiao, Mengyu Xu, Dongguang Fan, Ziwei Hu, Jiarui Wu, Tao Chen, Miao Liu, Xiaoguang Bao*, Hengte Ke*, andXingyue Ji*. A Bioorthogonal Decaging Chemistry of N-Oxide and Silylborane for Prodrug Activation both In Vitro and In Vivo. J. Am. Chem. Soc.2023, 145, 45, 24698–24706. (ACS Editors’ Choice)
Zhang Li, Yongming Wang, Miao Liu, Yiyao Pan, Zihui Ni, Qingqiang Min, Binghe Wang*, Hengte Ke*, and Xingyue Ji*. Reactive Oxygen Species-Activated Metal-Free Carbon Monoxide Prodrugs for Targeted Cancer Treatment. J. Med. Chem., 2023, 66, 14583–14596.
Qingqiang Min and Xingyue Ji*. Bioorthogonal Bond Cleavage Chemistry for On-demand Prodrug Activation: Opportunities and Challenges. J. Med. Chem. 2023, 66(24):16546-16567.
Shengchao Zhou, Kun Wang, Ziwei Hu, Tao Chen, Yao Dong, Rongmei Gao, Mengyuan Wu, Yuhuan Li, Xingyue Ji*. Design, synthesis, and structure-activity relationships of a novel class of quinazoline derivatives as coronavirus inhibitors. Eur. J. Med. Chem., 2023, 161, 115831.
Miao Liu, Zhang Li, Ziwei Hu, ZhiCheng Yan, Qingqiang Min, Wei Peng* and Xingyue Ji*. Dichloromethanol but not difluoromethanol as a viable surrogate of carbon monoxide for prodrug design. Chem. Commun., 2023, 59, 5583.
Ru Dong, Xiaoxiao Yang, Binghe Wang,* Xingyue Ji*. Mutual leveraging of proximity effects and click chemistry in chemical biology. Med. Res. Rev.2023, doi:10.1002/med.21927. (IF: 12.3)
Zhou Zhou, Shun Feng, Jujun Zhou, Xingyue Ji*, Ya-Qiu Long*. On-Demand Activation of a Bioorthogonal Prodrug of SN-38 with Fast Reaction Kinetics and High Releasing Efficiency In Vivo. J. Med. Chem.2022, 65(1):333-342. (IF: 8.0)
Qingqiang Min,# Zihui Ni,# Meng You, Miao Liu, Zhou Zhou, Hengte Ke*, Xingyue Ji*. Chemiexcitation-Triggered Prodrug Activation for Targeted Carbon Monoxide Delivery. Angew. Chem. Int. Ed.2022, 61, e202200974. (IF: 16.3)
Xingyue Ji*, Zhiyuan Zhong*. External stimuli-responsive gasotransmitter prodrugs: Chemistry and spatiotemporal release. J. Control. Release. 2022, 351, 81-101. (IF: 11.0)
2018.06-2020.06,四川大学华西医学院客座副教授;
JACS,Nature Communications, Science Translational Medicien,J. Med. Chem.,Advanced Science 等杂志审稿人。
气体信使小分子(CO, H2S等)药物化学生物学研究:发展新颖的脱笼(decaging)化学,用于气体信使小分子的可控靶向递送,并研究其在相关重大疾病的发生、发展以及治疗方面的作用。
新型Click化学的发现及其相关化学生物学研究:发展新颖的Click反应,并用于相关化学生物学研究,包括生物正交前药的设计,生物大分子的可逆可视化标记等。
抗感染、抗肿瘤靶向小分子药物的设计合成:基于传统药物化学策略,进行抗感染、抗肿瘤小分子靶向药物的设计与合成。
药学(药物化学)学硕,药学专硕,药学/化学生物学博士
Shunfei Cui, # Yiyao Pan, # Chenzhe Ma, Bin Qi, Qingqiang Min, Ming Li, Huabing Chen, * Hengte Ke,* and Xingyue Ji*. Self-assembled carbon monoxide nanoprodrug for chemiexcitation-triggered synergistic chemotherapy against breast cancer. Sci. China Chem., 2025, doi: 10.1007/s11426-024-2465-9.
Jiekai Sun, Xu Wang, Ye Gao, Shuangyu Li, Ziwei Hu, Yan Huang, Baoqiang Fan, Xia Wang, Miao Liu, Chunhua Qiao, Wei Zhang*, Yipeng Wang*, Xingyue Ji*. H2S scavenger as a broad-spectrum strategy to deplete bacteria-derived H2S for antibacterial sensitization. Nat. Commun., 2024, 15, 9422.
Zhicheng Yan, Yiyao Pan, Guofeng Jiao, Mengyu Xu, Dongguang Fan, Ziwei Hu, Jiarui Wu, Tao Chen, Miao Liu, Xiaoguang Bao*, Hengte Ke*, andXingyue Ji*. A Bioorthogonal Decaging Chemistry of N-Oxide and Silylborane for Prodrug Activation both In Vitro and In Vivo. J. Am. Chem. Soc.2023, 145, 45, 24698–24706. (ACS Editors’ Choice)
Zhang Li, Yongming Wang, Miao Liu, Yiyao Pan, Zihui Ni, Qingqiang Min, Binghe Wang*, Hengte Ke*, and Xingyue Ji*. Reactive Oxygen Species-Activated Metal-Free Carbon Monoxide Prodrugs for Targeted Cancer Treatment. J. Med. Chem., 2023, 66, 14583–14596.
Qingqiang Min and Xingyue Ji*. Bioorthogonal Bond Cleavage Chemistry for On-demand Prodrug Activation: Opportunities and Challenges. J. Med. Chem. 2023, 66(24):16546-16567.
Shengchao Zhou, Kun Wang, Ziwei Hu, Tao Chen, Yao Dong, Rongmei Gao, Mengyuan Wu, Yuhuan Li, Xingyue Ji*. Design, synthesis, and structure-activity relationships of a novel class of quinazoline derivatives as coronavirus inhibitors. Eur. J. Med. Chem., 2023, 161, 115831.
Miao Liu, Zhang Li, Ziwei Hu, ZhiCheng Yan, Qingqiang Min, Wei Peng* and Xingyue Ji*. Dichloromethanol but not difluoromethanol as a viable surrogate of carbon monoxide for prodrug design. Chem. Commun., 2023, 59, 5583.
Ru Dong, Xiaoxiao Yang, Binghe Wang,* Xingyue Ji*. Mutual leveraging of proximity effects and click chemistry in chemical biology. Med. Res. Rev.2023, doi:10.1002/med.21927. (IF: 12.3)
Zhou Zhou, Shun Feng, Jujun Zhou, Xingyue Ji*, Ya-Qiu Long*. On-Demand Activation of a Bioorthogonal Prodrug of SN-38 with Fast Reaction Kinetics and High Releasing Efficiency In Vivo. J. Med. Chem.2022, 65(1):333-342. (IF: 8.0)
Qingqiang Min,# Zihui Ni,# Meng You, Miao Liu, Zhou Zhou, Hengte Ke*, Xingyue Ji*. Chemiexcitation-Triggered Prodrug Activation for Targeted Carbon Monoxide Delivery. Angew. Chem. Int. Ed.2022, 61, e202200974. (IF: 16.3)
Xingyue Ji*, Zhiyuan Zhong*. External stimuli-responsive gasotransmitter prodrugs: Chemistry and spatiotemporal release. J. Control. Release. 2022, 351, 81-101. (IF: 11.0)
